Cell-penetrating pepducins targeting the neurotensin receptor type 1 relieve pain

Rebecca L. Brouillette, Élie Besserer-Offroy, Christine E. Mona +8

Pepducins are cell-penetrating, membrane-tethered lipopeptides designed to target the intracellular region of a G protein-coupled receptor (GPCR) in order to allosterically modulat…