72 citations · 123 across the 3 of their papers we have counts for
3 papers
Cell-penetrating pepducins targeting the neurotensin receptor type 1 relieve pain
Rebecca L. Brouillette, Élie Besserer-Offroy, Christine E. Mona +8
Pepducins are cell-penetrating, membrane-tethered lipopeptides designed to target the intracellular region of a G protein-coupled receptor (GPCR) in order to allosterically modulat…
The hypotensive effect of activated apelin receptor is correlated with \b{eta}-arrestin recruitment
Élie Besserer-Offroy, Patrick Bérubé, Jérôme Côté +8
The apelinergic system is an important player in the regulation of both vascular tone and cardiovascular function, making this physiological system an attractive target for drug de…
The signaling signature of the neurotensin type 1 receptor with endogenous ligands
Élie Besserer-Offroy, Rebecca L Brouillette, Sandrine Lavenus +8
The human neurotensin 1 receptor (hNTS1) is a G protein-coupled receptor involved in many physiological functions, including analgesia, hypothermia, and hypotension. To gain a bett…