activity
19982005
most citedDesign of HIV-1-PR inhibitors which do not create resistance: blocking the folding of single monomers

1 citations · 1 across the 2 of their papers we have counts for

collaborators

6 papers

q-bio.BM20051 cited

Design of HIV-1-PR inhibitors which do not create resistance: blocking the folding of single monomers

R. A. Broglia, G. Tiana, L. Sutto +2

One of the main problems of drug design is that of optimizing the drug--target interaction. In the case in which the target is a viral protein displaying a high mutation rate, a se…

cond-mat.soft2003

Understanding the determinants of stability and folding of small globular proteins from their energetics

G. Tiana, F. Simona, G. M. S. De Mori +2

The results of minimal model calculations suggest that the stability and the kinetic accessibility of the native state of small globular proteins are controlled by few "hot" sites.…

cond-mat.soft2002

Design and Folding of Dimeric Proteins

G. Tiana, R. A. Broglia

In a similar way in which the folding of single--domain proteins provide an important test in the study of self--organization, the folding of homodimers constitute a basic challeng…

cond-mat2000

Reading the three-dimensional structure of a protein from its amino acid sequence

R. A. Broglia, G. Tiana

While all the information required for the folding of a protein is contained in its amino acid sequence, one has not yet learnt how to extract this information so as to predict the…

cond-mat2000

Why does a protein fold?

R. A. Broglia, G. Tiana

With the help of lattice Monte Carlo modelling of heteropolymers, we show that the necessary condition for a protein to fold on short call is to proceed through partially folded in…

cond-mat.soft1998

Protein Foldability and Designability: General Physics and Pretty Chemistry

R. A. Broglia, G. Tiana, H. E. Roman

Making use of a simplified model for protein folding, it can be shown that conformations which are particularly stable when their energy is minimized with respect to amino acid seq…