18 citations · 36 across the 3 of their papers we have counts for
3 papers
A lipidated peptide derived from the C-terminal tail of the vasopressin 2 receptor shows promise as a new -arrestin inhibitor
Rebecca L. Brouillette, Christine E. Mona, Michael Desgagné +9
-arrestins play pivotal roles in seven transmembrane receptor (7TMR) signalling and trafficking. To study their functional role in the regulation of specific receptor systems, c…
Metabolically Stable Neurotensin Analogs Exert Potent and Long-Acting Analgesia Without Hypothermia
Mélanie Vivancos, Roberto Fanelli, Élie Besserer-Offroy +9
The endogenous tridecapeptide neurotensin (NT) has emerged as an important inhibitory modulator of pain transmission, exerting its analgesic action through the activation of the G…
Cell-penetrating pepducins targeting the neurotensin receptor type 1 relieve pain
Rebecca L. Brouillette, Élie Besserer-Offroy, Christine E. Mona +8
Pepducins are cell-penetrating, membrane-tethered lipopeptides designed to target the intracellular region of a G protein-coupled receptor (GPCR) in order to allosterically modulat…